Molecule Details
InChIKeyJTROLECZHRVLFM-UHFFFAOYSA-N
Compound Name7,8-dimethoxy-N-[1-(5-methyl-1H-pyrazol-3-yl)propan-2-yl]quinazolin-4-amine
Canonical SMILESCOc1ccc2c(NC(C)Cc3cc(C)[nH]n3)ncnc2c1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01064 PDE1B Homo sapiens Human PF00233 PF08499 7.7 IC50 ChEMBL;BindingDB
Q14123 PDE1C Homo sapiens Human PF00233 PF08499 7.1 IC50 ChEMBL;BindingDB
P54750 PDE1A Homo sapiens Human PF00233 PF08499 6.9 IC50 ChEMBL;BindingDB