Molecule Details
InChIKeyJTNXTIPDQKHRDT-VWLOTQADSA-N
Compound Nametert-butyl (2S)-2-[[[4-[4-[[1-[(4-fluoro-phenyl)carbamoyl]cyclo-propane-carbonyl]amino]phenoxy]-7-methoxyquinazoline-6-carbonyl]amino]methyl]pyr-rolidine-1-carboxylate
Canonical SMILESCOc1cc2ncnc(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3)c2cc1C(=O)NC[C@@H]1CCCN1C(=O)OC(C)(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.93
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30530 AXL Homo sapiens Human PF00041 PF13927 PF07714 7.3 IC50 BindingDB
Q12866 MERTK Homo sapiens Human PF00041 PF00047 PF13927 PF07714 7.3 IC50 BindingDB
P08581 MET Homo sapiens Human PF07714 PF01437 PF01403 PF01833 6.3 IC50 BindingDB