Molecule Details
InChIKeyJTNMHAMHIYAFAI-FQEVSTJZSA-N
Compound NameN-(4-{[3-Cyano-1-(2-methylpropyl)-1H-indazol-5-yl]oxy}phenyl)-L-prolinamide
Canonical SMILESCC(C)Cn1nc(C#N)c2cc(Oc3ccc(NC(=O)[C@@H]4CCCN4)cc3)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60825 PFKFB2 Homo sapiens Human PF01591 PF00300 7.8 IC50 ChEMBL;BindingDB
Q16875 PFKFB3 Homo sapiens Human PF01591 PF00300 7.5 IC50 ChEMBL;BindingDB
P16118 PFKFB1 Homo sapiens Human PF01591 PF00300 6.5 IC50 ChEMBL;BindingDB