Molecule Details
InChIKeyJTCNCYFBCGNCBJ-UHFFFAOYSA-N
Compound Name4-[[5-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]pyridin-2-yl]methyl]-1H-quinoxaline-2,3-dione
Canonical SMILESO=c1[nH]c2ccccc2n(Cc2ccc(-c3noc(C(F)(F)F)n3)cn2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 8.5 IC50 ChEMBL;BindingDB
Q9UQL6 HDAC5 Homo sapiens Human PF12203 PF00850 7.7 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 7.1 IC50 ChEMBL;BindingDB