Molecule Details
InChIKeyJSWXHRIKDWHCOW-UHFFFAOYSA-N
Compound Name3-amino-6-(2,6-difluorophenyl)-N-[4-(3-hydroxy-5-methylcyclohexen-1-yl)-3-pyridinyl]pyridine-2-carboxamide
Canonical SMILESCC1CC(c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)=CC(O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB