Molecule Details
InChIKeyJSRSTHPRYBNVDX-UHFFFAOYSA-N
Compound Name4-(1-benzofuran-2-yl)-2-[1-(3H-imidazo[4,5-c]pyridin-2-ylmethyl)piperidin-4-yl]-1,3-thiazole
Canonical SMILESc1ccc2oc(-c3csc(C4CCN(Cc5nc6cnccc6[nH]5)CC4)n3)cc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P10635 CYP2D6 Homo sapiens Human PF00067 6.3 IC50 ChEMBL;BindingDB
P10632 CYP2C8 Homo sapiens Human PF00067 6.2 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.1 IC50 ChEMBL;BindingDB