Molecule Details
InChIKeyJSPZPGCXQNWQIL-UHFFFAOYSA-N
Compound Name3-[2-[4-[4-fluoro-2-(2,2,2-trifluoroethoxy)phenyl]piperazin-1-yl]ethyl]-5-methyl-1H-pyrimidine-2,4-dione
Canonical SMILESCc1c[nH]c(=O)n(CCN2CCN(c3ccc(F)cc3OCC(F)(F)F)CC2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.3 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB