Molecule Details
InChIKeyJSCRCECGNHPGDY-UHFFFAOYSA-N
Compound NameN1-(2-(1-(6-carbamoylthieno[3,2-d]pyrimidin-4-yl)piperidin-4-yl)ethyl)-N3-ethylisophthalamide
Canonical SMILESCCNC(=O)c1cccc(C(=O)NCCC2CCN(c3ncnc4cc(C(N)=O)sc34)CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q8IXJ6 SIRT2 Homo sapiens Human PF02146 8.9 IC50 ChEMBL;BindingDB
Q9NTG7 SIRT3 Homo sapiens Human PF02146 8.3 IC50 ChEMBL;BindingDB
Q96EB6 SIRT1 Homo sapiens Human PF02146 8.3 IC50 ChEMBL;BindingDB