Molecule Details
InChIKeyJSBXKENODQYJRW-UHFFFAOYSA-N
Compound Name6-Hydroxy-benzothiazole-2-sulfonic acid [2-(N-methyl-guanidino)-acetyl]-amide
Canonical SMILESCN(CC(=O)NS(=O)(=O)c1nc2ccc(O)cc2s1)C(=N)N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.33
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.5 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.5 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 8.0 Ki ChEMBL;BindingDB