Molecule Details
InChIKeyJSBRNGDYGFBUPK-UHFFFAOYSA-N
Compound Name3-(aminomethyl)-4-(2,4-dichlorophenyl)-6-(4-methoxyphenyl)-2-methyl-5H-pyrrolo[3,4-b]pyridin-7-one
Canonical SMILESCOc1ccc(N2Cc3c(nc(C)c(CN)c3-c3ccc(Cl)cc3Cl)C2=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27487 DPP4 Homo sapiens Human PF00930 PF00326 8.0 Ki ChEMBL;BindingDB
Q6V1X1 DPP8 Homo sapiens Human PF19520 PF00930 PF00326 6.2 Ki ChEMBL;BindingDB
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 6.0 Ki ChEMBL;BindingDB