Molecule Details
InChIKeyJRVSGBSKZMZOOC-UHFFFAOYSA-N
Compound NameN-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]-N-[3-[(6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-yl)oxy]propyl]methanesulfonamide
Canonical SMILESCCCN1CCc2cccc3c2C1Cc1cccc(OCCCN(CCCN2CCN(c4ccccc4OC)CC2)S(C)(=O)=O)c1-3
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P21728 DRD1 Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB