Target not found.
Molecule Details
InChIKeyJRQYXWVDIBVRHN-UHFFFAOYSA-N
Compound NameN-tert-butyl-2-[3-[6-methyl-4-[4-(1H-pyrazol-4-yl)anilino]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]phenoxy]acetamide
Canonical SMILESCN1CCc2nc(-c3cccc(OCC(=O)NC(C)(C)C)c3)nc(Nc3ccc(-c4cn[nH]c4)cc3)c2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11166 SLC2A1 Homo sapiens Human PF00083 6.5 IC50 ChEMBL;BindingDB
P11169 SLC2A3 Homo sapiens Human PF00083 6.4 IC50 ChEMBL;BindingDB
O97467 ht1 Plasmodium falciparum Pathogen PF00083 6.8 IC50 ChEMBL;BindingDB