Molecule Details
InChIKeyJRPAZCAZXFNBAT-UHFFFAOYSA-N
Compound Name2-[4-[4-[2-(3-Fluoropropoxy)phenyl]piperazin-1-yl]butyl]-4-methyl-1,2,4-triazine-3,5-dione
Canonical SMILESCn1c(=O)cnn(CCCCN2CCN(c3ccccc3OCCCF)CC2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL7.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 6.5 Ki ChEMBL
P35348 ADRA1A Homo sapiens Human PF00001 6.5 Ki ChEMBL
P35368 ADRA1B Homo sapiens Human PF00001 6.5 Ki ChEMBL