Molecule Details
InChIKeyJRMVEEDZCPVFFK-UHFFFAOYSA-N
Compound Name9-chloro-3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2-methyl-7-(trifluoromethyl)pyrido[1,2-a]pyrimidin-4-one
Canonical SMILESCc1nc2c(Cl)cc(C(F)(F)F)cn2c(=O)c1CCN1CCc2oc3ccccc3c2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08913 ADRA2A Homo sapiens Human PF00001 8.9 IC50 ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P18825 ADRA2C Homo sapiens Human PF00001 8.4 IC50 ChEMBL;BindingDB