Molecule Details
InChIKeyJQWUZRQDRJVXDJ-UHFFFAOYSA-N
Compound Name(5-(Aminomethyl)-2-(8-methoxy-2-(trifluoromethyl)quinolin-5-yl)oxazol-4-yl)(4-(4,6-dimethoxypyrimidin-2-yl)piperazin-1-yl)methanone
Canonical SMILESCOc1cc(OC)nc(N2CCN(C(=O)c3nc(-c4ccc(OC)c5nc(C(F)(F)F)ccc45)oc3CN)CC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 8.7 IC50 ChEMBL;BindingDB
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 6.1 IC50 ChEMBL;BindingDB
Q9HCR9 PDE11A Homo sapiens Human PF01590 PF00233 6.0 IC50 ChEMBL;BindingDB