Molecule Details
InChIKeyJQUVQWMHZSYCRQ-UHFFFAOYSA-N
Canonical SMILESCCCCOc1c(OC)cc(C(=O)NCC2(N(C)C)CCOCC2)cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.06
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB16271
Drug NameOpiranserin
CAS Number1441000-45-8
Groups investigational
ATC Codes nan
DescriptionOpiranserin is under investigation in clinical trial NCT03997838 (Evaluate the Efficacy and Safety of VVZ-149 Injections for the Treatment of Post-operative Pain Following Abdominoplasty).

Cross-references: BindingDB: 50459963 CHEMBL4228903 ChemSpider: 64835236 Wikipedia: Opiranserin
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y345 SLC6A5 Homo sapiens Human PF00209 6.1 IC50 ChEMBL;BindingDB
P56373 P2RX3 Homo sapiens Human PF00864 6.1 IC50 ChEMBL