Molecule Details
InChIKeyJPIYOGKAIULUIO-UHFFFAOYSA-N
Compound Name5-(3,5-Difluoroanilino)pyrimido[4,5-c]quinoline-8-carboxylic acid
Canonical SMILESO=C(O)c1ccc2c(c1)nc(Nc1cc(F)cc(F)c1)c1ncncc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P68400 CSNK2A1 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P19784 CSNK2A2 Homo sapiens Human PF00069 8.1 IC50 ChEMBL
P67870 CSNK2B Homo sapiens Human PF01214 8.1 IC50 ChEMBL