Molecule Details
InChIKeyJPHBARUGZJTJNG-ZHRQHTTBSA-N
Compound NameN-[(4R,4aS,7R,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-dihydroxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]quinoline-3-carboxamide
Canonical SMILESO=C(N[C@@H]1CC[C@@]2(O)[C@H]3Cc4ccc(O)c5c4[C@@]2(CCN3CC2CC2)[C@H]1O5)c1cnc2ccccc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35372 OPRM1 Homo sapiens Human PF00001 10.2 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB