Molecule Details
InChIKeyJOSDAWJORYYQIX-UHFFFAOYSA-N
Compound Name4-(pyrazolo[1,5-b]pyridazin-3-yl)-N-(2,2,2-trifluoroethyl)pyrimidin-2-amine
Canonical SMILESFC(F)(F)CNc1nccc(-c2cnn3ncccc23)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.0
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 6.0 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 6.0 pIC50 TTD_MultiTarget