Molecule Details
InChIKeyJONJATYOSABZNY-UHFFFAOYSA-N
Compound Name7-cyclopentyl-2-[4-[2-(dimethylamino)ethylcarbamoyl]-2-fluoroanilino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide
Canonical SMILESCN(C)CCNC(=O)c1ccc(Nc2ncc3cc(C(=O)N(C)C)n(C4CCCC4)c3n2)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL8.38
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.6 IC50 ChEMBL
P30281 CCND3 Homo sapiens Human PF02984 PF00134 8.6 IC50 ChEMBL
O60563 CCNT1 Homo sapiens Human PF00134 PF21797 8.2 IC50 ChEMBL
P50750 CDK9 Homo sapiens Human PF00069 8.2 IC50 ChEMBL