Molecule Details
InChIKeyJOJOIJJNZOVEKT-UHFFFAOYSA-N
Compound Name3-[4-[[5-(1-Ethanimidoylpiperidin-4-yl)oxy-2-ethylbenzimidazol-1-yl]methyl]phenyl]benzenecarboximidamide
Canonical SMILESCCc1nc2cc(OC3CCN(C(C)=N)CC3)ccc2n1Cc1ccc(-c2cccc(C(=N)N)c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.8 Ki ChEMBL;BindingDB
P07477 PRSS1 Homo sapiens Human PF00089 6.8 Ki ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.7 Ki ChEMBL;BindingDB