Molecule Details
InChIKeyJOBHARMVZDXCRY-UHFFFAOYSA-N
Compound Name7,8-Dichloro-5-(4-chloro-phenyl)-2,5-dihydro-3H-imidazo[2,1-a]isoindol-5-ol
Canonical SMILESOC1(c2ccc(Cl)cc2)c2cc(Cl)c(Cl)cc2C2=NCCN21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01959 SLC6A3 Homo sapiens Human PF00209 8.6 IC50 ChEMBL;BindingDB
P23975 SLC6A2 Homo sapiens Human PF00209 7.7 IC50 ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 6.3 IC50 ChEMBL;BindingDB