Molecule Details
InChIKeyJNRTVZLIHFRYQO-UHFFFAOYSA-N
Compound NameN-(5-butyl-1,3-thiazol-2-yl)-6-methoxy-7-(3-morpholin-4-ylpropoxy)quinazolin-4-amine
Canonical SMILESCCCCc1cnc(Nc2ncnc3cc(OCCCN4CCOCC4)c(OC)cc23)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.22
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 8.2 pIC50 TTD_MultiTarget