Molecule Details
InChIKeyJNMYUIOIISURGX-MFCQPPMASA-N
Compound NameAc-Trp-Val-Thr-His-Cit-Leu-Ala-Gly-Leu-Leu-Ser-Cit-Ser-Gly-Gly-Val-Val-hArg-Lys-Asn-Phe-Val-Pro-Thr-Asp-Val-Gly-Oic(3axi,7axi)-Phe-Ala-Phe-NH2
Canonical SMILESCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](CCCNC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=O)C(=O)N[C@@H](CO)C(=O)NCC(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CCCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)NCC(=O)N1C2CCCCC2C[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1ccccc1)C(N)=O)C(C)C)[C@@H](C)O)C(C)C)C(C)C)C(C)C)[C@@H](C)O)C(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Unknown
Avg pChEMBL6.89
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P06881 CALCA Homo sapiens Human PF00214 8.7 IC50 ChEMBL;BindingDB
O60896 RAMP3 Homo sapiens Human PF04901 6.3 IC50 ChEMBL
Q16602 CALCRL Homo sapiens Human PF00002 PF02793 6.3 IC50 ChEMBL
Q7Z4H4 ADM2 Homo sapiens Human 6.3 IC50 BindingDB