Molecule Details
InChIKeyJLJLHTHYQPNRLZ-UHFFFAOYSA-N
Compound Name4-[6-methoxy-7-(2-piperidin-1-ylethoxy)quinazolin-4-yl]-N-(4-pyridin-2-ylphenyl)piperazine-1-carbothioamide
Canonical SMILESCOc1cc2c(N3CCN(/C(S)=N\c4ccc(-c5ccccn5)cc4)CC3)ncnc2cc1OCCN1CCCCC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.91
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q02161 RHD Homo sapiens Human PF00909 7.0 pIC50 TTD_MultiTarget
P09619 PDGFRB Homo sapiens Human PF00047 PF13927 PF25305 PF07714 6.8 IC50 ChEMBL;BindingDB