Molecule Details
InChIKeyJLIUDRVXSXMEGO-HHHXNRCGSA-N
Compound Name(4R)-3-acetyl-4-(3,4-difluorophenyl)-N-[3-[4-(4-fluorophenyl)piperidin-1-yl]propyl]-1,6-dimethyl-2-oxo-4H-pyrimidine-5-carboxamide
Canonical SMILESCC(=O)N1C(=O)N(C)C(C)=C(C(=O)NCCCN2CCC(c3ccc(F)cc3)CC2)[C@H]1c1ccc(F)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB