Molecule Details
InChIKeyJKPIUTPQBDXSRH-KYFHLAJPSA-N
Compound Name(2S,5R,8S,11R,14R)-8-[3-(diaminomethylideneamino)propyl]-2-(1H-imidazol-5-ylmethyl)-11-(1H-indol-3-ylmethyl)-5-(naphthalen-2-ylmethyl)-3,6,9,12,20,24-hexaoxo-1,4,7,10,13,19-hexazacyclotetracosane-14-carboxamide
Canonical SMILESN=C(N)NCCC[C@@H]1NC(=O)[C@@H](Cc2ccc3ccccc3c2)NC(=O)[C@H](Cc2c[nH]cn2)NC(=O)CCCC(=O)NCCCC[C@H](C(N)=O)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41968 MC3R Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB