Molecule Details
InChIKeyJKJKHYOUTNOITO-KEJHGIAHSA-N
Compound Name(3S)-3-[[(3S)-3-[[2-[(2S)-1-[2-[(2S)-1-[(4R,10R,13S,16S,19S,22R,25S)-25-acetyl-22-(2-carboxyethyl)-13-[3-(diaminomethylideneamino)propyl]-19-(1H-imidazol-4-ylmethyl)-10-(1H-indol-3-ylmethyl)-16-(naphthalen-2-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptazacyclohexacosane-4-carbonyl]pyrrolidin-2-yl]-2-oxoethyl]pyrrolidin-2-yl]-2-oxoethyl]amino]-7-amino-2-oxoheptyl]amino]-4-amino-4-oxobutanoic acid
Canonical SMILESCC(=O)[C@@H]1CSSC[C@@H](C(=O)N2CCC[C@H]2C(=O)CN2CCC[C@H]2C(=O)CN[C@@H](CCCCN)C(=O)CN[C@@H](CC(=O)O)C(N)=O)NC(=O)CNC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc2ccc3ccccc3c2)NC(=O)[C@H](Cc2c[nH]cn2)NC(=O)[C@@H](CCC(=O)O)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 7.4 IC50 ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB