Molecule Details
InChIKeyJKHGXFOISOLZKF-UHFFFAOYSA-N
Compound Name6-chloro-N-[2,4-difluoro-5-[5-(2,4,5-trifluoro-3-hydroxybenzoyl)thiophen-2-yl]phenyl]pyridine-3-sulfonamide
Canonical SMILESO=C(c1ccc(-c2cc(NS(=O)(=O)c3ccc(Cl)nc3)c(F)cc2F)s1)c1cc(F)c(F)c(O)c1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P37059 HSD17B2 Homo sapiens Human PF00106 8.5 IC50 ChEMBL;BindingDB
P14061 HSD17B1 Homo sapiens Human PF00106 8.1 IC50 ChEMBL;BindingDB