Molecule Details
InChIKeyJKGFOIGGPUTHIY-UHFFFAOYSA-N
Compound Name2,2-Dimethyl-5-morpholino-N-(pyridin-3-ylmethyl)-2,4-dihydro-1H-pyrano[4'',3'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-8-amine
Canonical SMILESCC1(C)Cc2c(c(N3CCOCC3)nc3sc4c(NCc5cccnc5)ncnc4c23)CO1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 8.2 IC50 ChEMBL;BindingDB
P27815 PDE4A Homo sapiens Human PF18100 PF00233 7.3 IC50 ChEMBL;BindingDB
Q08499 PDE4D Homo sapiens Human PF18100 PF00233 7.3 IC50 ChEMBL;BindingDB