Molecule Details
InChIKeyJKFGTURSEBTJIZ-UHFFFAOYSA-N
Compound Name4-(5-chloro-3-isopropyl-1H-pyrazol-4-yl)-N-(5-(4-(dimethylamino)piperidin-1-yl)pyridin-2-yl)pyrimidin-2-amine
Canonical SMILESCC(C)c1n[nH]c(Cl)c1-c1ccnc(Nc2ccc(N3CCC(N(C)C)CC3)cn2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.0
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.0 pIC50 TTD_MultiTarget
P24385 CCND1 Homo sapiens Human PF02984 PF00134 8.0 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 8.0 pIC50 TTD_MultiTarget