Molecule Details
InChIKeyJJQLRTKUCLCIPR-UHFFFAOYSA-N
Compound Name4-Bromo-N-[4-(quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide
Canonical SMILESO=S(=O)(NC1CCC(Nc2ncc3ccccc3n2)CC1)c1ccc(Br)cc1OC(F)(F)F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08913 ADRA2A Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB
Q99705 MCHR1 Homo sapiens Human PF00001 7.1 IC50 ChEMBL;BindingDB
Q15761 NPY5R Homo sapiens Human PF00001 6.1 IC50 ChEMBL;BindingDB