Molecule Details
InChIKeyJJEUGQSNWGGUIG-SFTDATJTSA-N
Compound Name1-phenyl-4-[(11S,16R)-6-thia-10,14-diazatetracyclo[8.6.1.05,17.011,16]heptadeca-1(17),2,4-trien-14-yl]butan-1-one
Canonical SMILESO=C(CCCN1CC[C@H]2[C@@H](C1)c1cccc3c1N2CCCS3)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB