Molecule Details
InChIKeyJIQRMBNAYWCUEG-UHFFFAOYSA-N
Compound NameN-[5-bromo-6-(4-hydroxyphenyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]-4-(4-ethylpiperazin-1-yl)butanamide
Canonical SMILESCCN1CCN(CCCC(=O)Nc2n[nH]c3nc(-c4ccc(O)cc4)c(Br)cc23)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.01
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49840 GSK3A Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB