Molecule Details
InChIKeyJINXSJRUNKRAKJ-UHFFFAOYSA-N
Compound NameN-[5-[(4-ethylpiperazin-1-yl)methyl]pyrazin-2-yl]-6-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-4-amine
Canonical SMILESCCN1CCN(Cc2cnc(Nc3cc(-c4cc(F)c5nc(C)n(C(C)C)c5c4)ncn3)cn2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.09
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 8.6 IC50 ChEMBL;BindingDB
P06493 CDK1 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB