Molecule Details
InChIKeyJICSVJQEGDFDBH-ULNSLHSMSA-N
Compound Name(S)-2-((S)-4-((R)-3-(4-Fluorophenyl)-2-(2-(methylamino)acetamido)propanoyl)-2-oxo-3-propylpiperazin-1-yl)-N-methyl-3-(naphthalen-2-yl)propanamide
Canonical SMILESCCC[C@H]1C(=O)N([C@@H](Cc2ccc3ccccc3c2)C(=O)NC)CCN1C(=O)[C@@H](Cc1ccc(F)cc1)NC(=O)CNC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.14
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
Q01726 MC1R Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB