Molecule Details
InChIKeyJHWYFIOMMXUNLT-UHFFFAOYSA-N
Compound Name2-amino-7-fluoro-N-(quinolin-8-ylmethyl)quinazoline-4-carboxamide
Canonical SMILESNc1nc(C(=O)NCc2cccc3cccnc23)c2ccc(F)cc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.52
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.5 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB