Molecule Details
InChIKeyJHVGQSBTPJECOW-UHFFFAOYSA-N
Compound Name1-(3-Chlorophenyl)sulfonyl-2-phenyl-4-piperazin-1-ylimidazo[4,5-c]pyridine
Canonical SMILESO=S(=O)(c1cccc(Cl)c1)n1c(-c2ccccc2)nc2c(N3CCNCC3)nccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P50406 HTR6 Homo sapiens Human PF00001 7.9 IC50 ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB