Molecule Details
InChIKeyJGRMMBRYUDVUAI-UHFFFAOYSA-N
Compound Name8-Fluoro-6-Methoxy-3,4-Dimethyl-1-(3-Methylpyridin-4-Yl)imidazo[1,5-A]quinoxaline
Canonical SMILESCOc1cc(F)cc2c1nc(C)c1c(C)nc(-c3ccncc3C)n12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.65
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 9.2 IC50 ChEMBL;BindingDB
O00408 PDE2A Homo sapiens Human PF01590 PF00233 7.0 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.8 IC50 ChEMBL;BindingDB