Molecule Details
InChIKeyJGESVFFMSKZGDK-UHFFFAOYSA-N
Compound Name4-(4-chlorophenoxy)-N-(1-hydroxy-2-oxo-3-pyridinyl)-N-[2-(4-methylpiperazin-1-yl)ethyl]benzenesulfonamide
Canonical SMILESCN1CCN(CCN(c2cccn(O)c2=O)S(=O)(=O)c2ccc(Oc3ccc(Cl)cc3)cc2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.83
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.9 IC50 ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.8 pIC50 TTD_MultiTarget