Molecule Details
InChIKeyJFWOCEJLRQNSEH-GFCCVEGCSA-N
Compound Name2-[(2R)-2-(pyridin-3-yloxymethyl)piperazin-1-yl]-[1,3]oxazolo[4,5-b]pyridine
Canonical SMILESc1cncc(OC[C@H]2CNCCN2c2nc3ncccc3o2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36544 CHRNA7 Homo sapiens Human PF02931 PF02932 8.2 IC50 ChEMBL;BindingDB
P17787 CHRNB2 Homo sapiens Human PF02931 PF02932 7.2 IC50 ChEMBL
P43681 CHRNA4 Homo sapiens Human PF02931 PF02932 7.2 IC50 ChEMBL;BindingDB