Molecule Details
InChIKeyJFSBDKASCAKCDV-MUGJNUQGSA-N
Compound Name(S)-2-[(2-{(S)-2-[((R)-2-Amino-3-mercapto-propionyl)-methyl-amino]-3-methyl-butyryl}-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl)-amino]-4-methylsulfanyl-butyric acid
Canonical SMILESCSCC[C@H](NC(=O)[C@@H]1Cc2ccccc2CN1C(=O)[C@H](C(C)C)N(C)C(=O)[C@@H](N)CS)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.3
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.3 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.3 IC50 ChEMBL;BindingDB