Molecule Details
InChIKeyJFRTUZNKHJJSEH-AWEZNQCLSA-N
Compound Name3-[(3S)-3-amino-1-piperidyl]-5-[6-(6-methylpyrazin-2-yl)pyrazolo[4 3-c]pyridin-1-yl]pyrazin-2-ol
Canonical SMILESCc1cncc(-c2cc3c(cn2)cnn3-c2cnc(O)c(N3CCC[C@H](N)C3)n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.5
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.7 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.6 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.2 Ki ChEMBL;BindingDB