Molecule Details
InChIKeyJFRJCQJVFMHZOO-QZHHGCDDSA-N
Compound NameN-(2-Aminoethyl)-2-(4-(2-(4-((9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-9H-purin-6-yl)amino)phenyl)acetamido)phenyl)acetamide
Canonical SMILESNCCNC(=O)Cc1ccc(NC(=O)Cc2ccc(Nc3ncnc4c3ncn4[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)cc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.44
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P0DMS8 ADORA3 Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB