Molecule Details
InChIKeyJFJRYQOFIDFJKY-UHFFFAOYSA-N
Compound Name2-{[2-({1-[2-(dimethylamino)acetyl]-6-methoxy-1,2,3,4-tetrahydroquinolin-7-yl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-6-fluorobenzamide
Canonical SMILESCOc1cc2c(cc1Nc1nc(Nc3cccc(F)c3C(N)=O)c3cc[nH]c3n1)N(C(=O)CN(C)C)CCC2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.0
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06729 CD2 Homo sapiens Human PF05790 PF07686 9.0 pIC50 TTD_MultiTarget
P08069 IGF1R Homo sapiens Human PF00757 PF07714 PF01030 9.0 IC50 ChEMBL;BindingDB