Molecule Details
InChIKeyJFHRDTICJOZJOB-UHFFFAOYSA-N
Canonical SMILESCCOc1cc(C(=O)NC2CC2)cc(-c2cccc(-c3cc(NC(=O)Nc4c(Cl)cncc4Cl)c(=O)n(CC)n3)c2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.37
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 9.5 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB