Molecule Details
InChIKeyJEZKKPXWSVQUPH-NBGIEHNGSA-N
Compound Name(1S,2R)-1-(3,4-dichlorophenyl)-2-((4-(N,N-dimethylsulfamoyl)piperazin-1-yl)methyl)-N-(4-fluorobenzyl)-N-methylcyclopropanecarboxamide
Canonical SMILESCN(Cc1ccc(F)cc1)C(=O)[C@@]1(c2ccc(Cl)c(Cl)c2)C[C@H]1CN1CCN(S(=O)(=O)N(C)C)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29371 TACR3 Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P21452 TACR2 Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB
P25103 TACR1 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB