Molecule Details
InChIKeyJEHBCDCKKVKVGB-UHFFFAOYSA-N
Compound NameUS9751837, Example 19
Canonical SMILESCOc1cc(Nc2cc(Oc3ccc(NC(=O)Nc4cc(C(C)(C)C)cc(NS(C)(=O)=O)c4OC)c4ccccc34)ccn2)ccc1C(=O)NCCOCCCOCOP(=O)(O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43405 SYK Homo sapiens Human PF07714 PF00017 8.1 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 7.7 IC50 ChEMBL;BindingDB