Molecule Details
InChIKeyJEBJXGHLBZQKNY-UHFFFAOYSA-N
Compound Name5-(4-(4-Chlorophenyl)-5-(1,5-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)-6-oxo-1-propyl-1,4,5,6-tetrahydropyrrolo[3,4-d]imidazol-2-yl)nicotinonitrile
Canonical SMILESCCCn1c(-c2cncc(C#N)c2)nc2c1C(=O)N(c1cc(C)c(=O)n(C)c1)C2c1ccc(Cl)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 6.8 IC50 ChEMBL;BindingDB
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 6.8 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 6.6 IC50 ChEMBL;BindingDB