Molecule Details
InChIKeyJDQOICVJUDEXEQ-UHFFFAOYSA-N
Canonical SMILESCN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C(=O)c1c(OCCCC2CCN(C(=O)OC3(C)CC3)CC2)c2ccccc2n(C)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q8NHU3 SGMS2 Homo sapiens Human PF14360 7.5 Kd ChEMBL;BindingDB
Q86VZ5 SGMS1 Homo sapiens Human PF14360 6.0 IC50 ChEMBL;BindingDB